^Thanawala, V.; Kadam, V.; Ghosh, R. (1 October 2008). "Enkephalinase Inhibitors: Potential Agents for the Management of Pain". Current Drug Targets. 9 (10): 887–894. doi:10.2174/138945008785909356. PMID 18855623.
^Noble, Florence; Roques, Bernard P (17 January 2007). "Protection of endogenous enkephalin catabolism as natural approach to novel analgesic and antidepressant drugs". Expert Opinion on Therapeutic Targets. 11 (2): 145–159. doi:10.1517/14728222.11.2.145. PMID 17227231. S2CID 24437682.
May 03, 2024
3007, orally, active, analogue, acts, enkephalinase, inhibitor, which, used, scientific, research, names, iupac, name, benzyl, acetylsulfanyl, ethoxy, amino, phenyl, methyl, phosphonoyl, methyl, biphenyl, propanoyl, alaninate, systematic, iupac, name, benzyl, . RB 3007 is an orally active analogue of RB 101 It acts as an enkephalinase inhibitor which is used in scientific research 1 2 RB 3007 Names IUPAC name Benzyl N 2S 2 2 acetylsulfanyl ethoxy R amino phenyl methyl phosphonoyl methyl 3 1 1 biphenyl 4 yl propanoyl L alaninate Systematic IUPAC name Benzyl 9S 12S 7 R amino phenyl methyl 9 1 1 biphenyl 4 yl methyl 12 methyl 2 7 10 trioxo 6 oxa 3 thia 11 aza 7l5 phosphatridecan 13 oate Other names RB3007 LS 15768 Identifiers 3D model JSmol Interactive image ChemSpider 9247929 PubChem CID 11072779 InChI InChI 1S C37H41N2O6PS c1 27 37 42 44 25 30 12 6 3 7 13 30 39 36 41 34 24 29 18 20 32 21 19 29 31 14 8 4 9 15 31 26 46 43 45 22 23 47 28 2 40 35 38 33 16 10 5 11 17 33 h3 21 27 34 35H 22 26 38H2 1 2H3 H 39 41 t27 34 35 46 m0 s1Key PYJMLILRVYLUHW UNCDKACKSA N SMILES C C H NC O C H CC1 CC C C C1 C1 CC CC C1 CP O OCCSC C O C H N C1 CC CC C1 C O OCC1 CC CC C1 Properties Chemical formula C 37H 41N 2O 6P S Molar mass 672 78 g mol 1 Except where otherwise noted data are given for materials in their standard state at 25 C 77 F 100 kPa Infobox referencesSee also editRB 101 enkephalinase inhibitor that produces analgesia without respiratory depression D DL Phenylalanine D phenylalanine blockage of enkephalin degradation may be responsible for the reputed analgesic effect of DL Phenylalanine Racecadotril an antidiarrheal drug which acts as a peripheral enkephalinase inhibitor Ecadotril a neutral endopeptidase inhibitorReferences edit Thanawala V Kadam V Ghosh R 1 October 2008 Enkephalinase Inhibitors Potential Agents for the Management of Pain Current Drug Targets 9 10 887 894 doi 10 2174 138945008785909356 PMID 18855623 Noble Florence Roques Bernard P 17 January 2007 Protection of endogenous enkephalin catabolism as natural approach to novel analgesic and antidepressant drugs Expert Opinion on Therapeutic Targets 11 2 145 159 doi 10 1517 14728222 11 2 145 PMID 17227231 S2CID 24437682 Retrieved from https en wikipedia org w index php title RB 3007 amp oldid 1153522446, wikipedia, wiki, book, books, library,
