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List of antiretroviral fixed-dose combinations

Antiretroviral drugs are used to manage HIV/AIDS. Multiple antiretroviral drugs are often combined into a single pill in order to reduce pill burden.

Some of these combinations are complete single-tablet regimens; the others must be combined with additional pills to make a treatment regimen.

Brand name(s) Ingredients (INN) Food and Drug Administration (FDA) approval date European Medicines Agency (EMA) approval date Health Canada approval date Company Single-tablet regimen?
NRTIs / NtRTIs NNRTI INSTI PI PK enhancer
Combivir lamivudine
zidovudine
September 26, 1997 ViiV Healthcare No
Kaletra (developed countries)
Aluvia (developing countries)
lopinavir ritonavir September 15, 2000 Abbott Laboratories No
Trizivir abacavir
lamivudine
zidovudine
November 15, 2000 ViiV Healthcare Yes
Epzicom (US)
Kivexa (EU, RU)
abacavir
lamivudine
August 2, 2004 ViiV Healthcare No
Generics, e.g., Triomune lamivudine
stavudine
nevirapine (not approved) (many companies) Yes
Generics, e.g., Duovir-N lamivudine
zidovudine
nevirapine (not approved) (many companies) Yes
Truvada emtricitabine
tenofovir disoproxil
August 2, 2004 Gilead Sciences No
Atripla emtricitabine
tenofovir disoproxil
efavirenz July 12, 2006 Gilead Sciences
Bristol-Myers Squibb
Yes
Complera (US)
Eviplera (EU, RU)
emtricitabine
tenofovir disoproxil
rilpivirine August 10, 2011 Gilead Sciences
Janssen Pharmaceutica
Yes
Stribild emtricitabine
tenofovir disoproxil
elvitegravir cobicistat August 27, 2012 Gilead Sciences Yes
Triumeq abacavir
lamivudine
dolutegravir August 22, 2014 ViiV Healthcare Yes
Evotaz atazanavir cobicistat January 29, 2015 Bristol-Myers Squibb No
Prezcobix (US)
Rezolsta (EU)
darunavir cobicistat January 29, 2015 Janssen Pharmaceutica No
Dutrebis lamivudine raltegravir February 6, 2015 Merck & Co. No
Genvoya emtricitabine
tenofovir alafenamide
elvitegravir cobicistat November 5, 2015 Gilead Sciences Yes
Odefsey emtricitabine
tenofovir alafenamide
rilpivirine March 1, 2016 Gilead Sciences Yes
Descovy emtricitabine
tenofovir alafenamide
April 4, 2016 Gilead Sciences No
Juluca rilpivirine dolutegravir November 21, 2017 ViiV Healthcare Yes
Symfi, Symfi Lo lamivudine
tenofovir disoproxil
efavirenz February 5, 2018 (Symfi Lo)
March 22, 2018 (Symfi)
Mylan Yes
Biktarvy emtricitabine
tenofovir alafenamide
bictegravir February 7, 2018 Gilead Sciences Yes
Cimduo, Temixys lamivudine
tenofovir disoproxil
February 28, 2018 Mylan No
Symtuza emtricitabine
tenofovir alafenamide
darunavir cobicistat July 17, 2018 Janssen Pharmaceutica Yes
Delstrigo lamivudine
tenofovir disoproxil
doravirine August 30, 2018 Merck & Co. Yes
Dovato lamivudine dolutegravir April 8, 2019 ViiV Healthcare Yes
Cabenuva rilpivirine cabotegravir January 21, 2021 March 18, 2020[1][2] ViiV Healthcare No

References edit

  1. ^ "Cabenuva Product information". Health Canada. 25 April 2012. Retrieved 22 January 2021.
  2. ^ "ViiV Healthcare announces first global regulatory approval of Cabenuva; the first complete, long-acting, regimen for the treatment of HIV". GSK. Retrieved 23 January 2021.

External links edit

  • "Appendix A, Table 1. Antiretrovirals Available in Fixed-Dose Combination Tablets". ClinicalInfo.   This article incorporates text from this source, which is in the public domain.

list, antiretroviral, fixed, dose, combinations, this, article, needs, additional, citations, verification, please, help, improve, this, article, adding, citations, reliable, sources, unsourced, material, challenged, removed, find, sources, news, newspapers, b. This article needs additional citations for verification Please help improve this article by adding citations to reliable sources Unsourced material may be challenged and removed Find sources List of antiretroviral fixed dose combinations news newspapers books scholar JSTOR January 2021 Learn how and when to remove this message Antiretroviral drugs are used to manage HIV AIDS Multiple antiretroviral drugs are often combined into a single pill in order to reduce pill burden Some of these combinations are complete single tablet regimens the others must be combined with additional pills to make a treatment regimen Brand name s Ingredients INN Food and Drug Administration FDA approval date European Medicines Agency EMA approval date Health Canada approval date Company Single tablet regimen NRTIs NtRTIs NNRTI INSTI PI PK enhancer Combivir lamivudinezidovudine September 26 1997 ViiV Healthcare No Kaletra developed countries Aluvia developing countries lopinavir ritonavir September 15 2000 Abbott Laboratories No Trizivir abacavirlamivudinezidovudine November 15 2000 ViiV Healthcare Yes Epzicom US Kivexa EU RU abacavirlamivudine August 2 2004 ViiV Healthcare No Generics e g Triomune lamivudinestavudine nevirapine not approved many companies Yes Generics e g Duovir N lamivudinezidovudine nevirapine not approved many companies Yes Truvada emtricitabinetenofovir disoproxil August 2 2004 Gilead Sciences No Atripla emtricitabinetenofovir disoproxil efavirenz July 12 2006 Gilead SciencesBristol Myers Squibb Yes Complera US Eviplera EU RU emtricitabinetenofovir disoproxil rilpivirine August 10 2011 Gilead SciencesJanssen Pharmaceutica Yes Stribild emtricitabinetenofovir disoproxil elvitegravir cobicistat August 27 2012 Gilead Sciences Yes Triumeq abacavirlamivudine dolutegravir August 22 2014 ViiV Healthcare Yes Evotaz atazanavir cobicistat January 29 2015 Bristol Myers Squibb No Prezcobix US Rezolsta EU darunavir cobicistat January 29 2015 Janssen Pharmaceutica No Dutrebis lamivudine raltegravir February 6 2015 Merck amp Co No Genvoya emtricitabinetenofovir alafenamide elvitegravir cobicistat November 5 2015 Gilead Sciences Yes Odefsey emtricitabinetenofovir alafenamide rilpivirine March 1 2016 Gilead Sciences Yes Descovy emtricitabinetenofovir alafenamide April 4 2016 Gilead Sciences No Juluca rilpivirine dolutegravir November 21 2017 ViiV Healthcare Yes Symfi Symfi Lo lamivudinetenofovir disoproxil efavirenz February 5 2018 Symfi Lo March 22 2018 Symfi Mylan Yes Biktarvy emtricitabinetenofovir alafenamide bictegravir February 7 2018 Gilead Sciences Yes Cimduo Temixys lamivudinetenofovir disoproxil February 28 2018 Mylan No Symtuza emtricitabinetenofovir alafenamide darunavir cobicistat July 17 2018 Janssen Pharmaceutica Yes Delstrigo lamivudinetenofovir disoproxil doravirine August 30 2018 Merck amp Co Yes Dovato lamivudine dolutegravir April 8 2019 ViiV Healthcare Yes Cabenuva rilpivirine cabotegravir January 21 2021 March 18 2020 1 2 ViiV Healthcare NoReferences edit Cabenuva Product information Health Canada 25 April 2012 Retrieved 22 January 2021 ViiV Healthcare announces first global regulatory approval of Cabenuva the first complete long acting regimen for the treatment of HIV GSK Retrieved 23 January 2021 External links edit Appendix A Table 1 Antiretrovirals Available in Fixed Dose Combination Tablets ClinicalInfo nbsp This article incorporates text from this source which is in the public domain Portals nbsp Medicine nbsp Viruses Retrieved from https en wikipedia org w index php title List of antiretroviral fixed dose combinations amp oldid 1205419457, wikipedia, wiki, book, books, library,

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